77-301-0
Tocris Bioscience™ AS2717638
Manufacturer: Tocris Bioscience™
CAS Number: 2148339-28-8
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 77-301-0-Each-of-1 | In Stock | ₹ 27,323.00 |
77-301-0 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 27,323.00
GST (18%): ₹ 4,918.14
Total Price: ₹ 32,241.14
Chemical Name or Material
6,7-Dimethoxy-2-(5-methyl-1,2-benzisoxazol-3-yl)-4-(1-piperidinylcarbonyl)-1(2 H)-isoquinolinone
Quantity
10 mg
Molecular Formula
C25H25N3O5
CAS
2148339-28-8
Target
LPAR5/LPA5/GPR92
Purity
0.98
Other Options
| Image | Product Name | Manufacturer | Price Range | |
|---|---|---|---|---|
 | Medchemexpress LLC HY-114379 5mg Medchemexpress, AS2717638 CAS:2148339-28-8 Purity:>98% | Medchemexpress LLC | ₹ 36,445.50 | |
 | 2148339-28-8 | AS2717638 | A2B Chem | ₹ 5,785.00 - ₹ 99,324.00 |
Related Products
Description
- AS2717638 is a potent LPA5 receptor antagonist (IC50 = 38 nM in BV-2 microglia cells)
- It is selective for LPA5 over LPA1, LPA2, and LPA3
- It inhibits LPA-mediated pro-inflammatory transcription factor phosphorylation
- In vivo , AS2717638 inhibits LPA5 agonist-induced allodynia in mice
- It also exhibits analgesic effects against both neuropathic and inflammatory pain in rodent models
- Orally bioavailable and brain penetrant.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
Compare Similar Items
Show Difference
Chemical Name or Material: 6,7-Dimethoxy-2-(5-methyl-1,2-benzisoxazol-3-yl)-4-(1-piperidinylcarbonyl)-1(2 H)-isoquinolinone
Quantity: 10 mg
Molecular Formula: C25H25N3O5
CAS: 2148339-28-8
Target: LPAR5/LPA5/GPR92
Purity: 0.98
Chemical Name or Material:
6,7-Dimethoxy-2-(5-methyl-1,2-benzisoxazol-3-yl)-4-(1-piperidinylcarbonyl)-1(2 H)-isoquinolinone
Quantity:
10 mg
Molecular Formula:
C25H25N3O5
CAS:
2148339-28-8
Target:
LPAR5/LPA5/GPR92
Purity:
0.98
Chemical Name or Material: Methyl (2S)-2-[[(4-methylphenyl)sulfonyl]amino]-9,13-dioxo-14-phenyl-7-[[[[(2-phenylacetyl)oxy]methoxy]carbonyl]amino]-10,12-dioxa-6,8-diazatetradec-6-enoate
Quantity: 1 mg
Molecular Formula: C34H38N4O12S
CAS: 1362911-19-0
Target: APC
Purity: 90%
Chemical Name or Material:
Methyl (2S)-2-[[(4-methylphenyl)sulfonyl]amino]-9,13-dioxo-14-phenyl-7-[[[[(2-phenylacetyl)oxy]methoxy]carbonyl]amino]-10,12-dioxa-6,8-diazatetradec-6-enoate
Quantity:
1 mg
Molecular Formula:
C34H38N4O12S
CAS:
1362911-19-0
Target:
APC
Purity:
90%
Chemical Name or Material: 5-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride
Quantity: 25 mg
Molecular Formula: C17H20N4O5.HCl
CAS: __
Target: CRBN
Purity: 0.95
Chemical Name or Material:
5-[(2-(2-Aminoethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride
Quantity:
25 mg
Molecular Formula:
C17H20N4O5.HCl
CAS:
__
Target:
CRBN
Purity:
0.95
Chemical Name or Material: 5-[(2-(2-(2-Aminoethoxy)ethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride
Quantity: 25 mg
Molecular Formula: C19H24N4O6.HCl
CAS: 2357110-58-6
Target: CRBN
Purity: 0.95
Chemical Name or Material:
5-[(2-(2-(2-Aminoethoxy)ethoxy)ethyl)amino]-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride
Quantity:
25 mg
Molecular Formula:
C19H24N4O6.HCl
CAS:
2357110-58-6
Target:
CRBN
Purity:
0.95