7112433

Tocris Bioscience™ TASP 0390325

Potent and selective V1B receptor antagonist; orally bioavailable

Manufacturer: Fischer Scientific

CAS Number: 1642187-96-9

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Product Type

Antagonist

CAS

1642187-96-9

Formula Weight

554.44g/mol

For Use With (Application)

Vasopressin Receptor Antagonists

Target Proteins

Vasopressin Receptor

Molecular Formula

C25H29ClFN5O4.HCl

Content And Storage

Store at -20°C

Other Options

Image Product Name Manufacturer Price Range
57-291-0
Tocris Bioscience™ TASP 0390325
Fischer Scientific ₹ 27,892.56
57-295-0
Tocris Bioscience™ TASP 0390325
Fischer Scientific ₹ 1,15,848.24
AX63118
1642187-96-9 | 2-(2-(3-Chloro-4-fluorophenyl)-6-(3-morpholinopropoxy)-4-oxopyrido[2,3-d]pyrimidin-3(4H)-yl)-N-isopropylacetamide hydroChloride
A2B Chem ₹ 16,513.08 - ₹ 1,42,286.28

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Description

  • Potent and selective V1B receptor antagonist (IC50 = 2.22 nM for rat pituitary receptor)
  • Exhibits no significant affinity for 85 other receptors, ion channels and transporters at 10 μM, including V1A and V2
  • Increases ACTH levels in rats
  • Orally bioavailable
  • Antidepressant and anxiolytic.

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Product Type:
Antagonist

CAS:
1642187-96-9

Formula Weight:
554.44g/mol

For Use With (Application):
Vasopressin Receptor Antagonists

Target Proteins:
Vasopressin Receptor

Molecular Formula:
C25H29ClFN5O4.HCl

Content And Storage:
Store at -20°C

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Molecular Formula:
C15H14ClFN4O2S2

Content And Storage:
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Formula Weight:
626.62g/mol

For Use With (Application):
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Molecular Formula:
C31H32BrNO4S2

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