70-291-0
Tocris™ GX 201
Manufacturer: Tocris™
CAS Number: 1788071-27-1
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 70-291-0-Each-of-1 | In Stock | ₹ 33,411.18 |
70-291-0 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 33,411.18
GST (18%): ₹ 6,014.012
Total Price: ₹ 39,425.192
Chemical Name or Material
4-[[1-[[2-Chloro-5-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methoxy]-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide
Quantity
10 mg
Molecular Formula
C25H27ClF4N2O4S
CAS
1788071-27-1
Target
Voltage-gated Sodium Channel Blockers
Purity
0.98
Related Products
Description
- GX 201 is a potent and selective Nav1.7 blocker (IC50 = 3.2 nM)
- Exhibits 10x selectivity for Nav1.7 over Nav1.1, Nav1.2, and Nav1.6 channels
- Displays prolonged residency time on the Nav1.7 channel
- Chronic dosing increases compound potency ∽10-fold and provides efficacy that persists after the compound has cleared from plasma
- Suppresses neuropathic pain in a mouse diabetic neuropathy model
- Analgesic.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
Compare Similar Items
Show Difference
Chemical Name or Material: 4-[[1-[[2-Chloro-5-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methoxy]-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide
Quantity: 10 mg
Molecular Formula: C25H27ClF4N2O4S
CAS: 1788071-27-1
Target: Voltage-gated Sodium Channel Blockers
Purity: 0.98
Chemical Name or Material:
4-[[1-[[2-Chloro-5-(trifluoromethyl)phenyl]methyl]-4-piperidinyl]methoxy]-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide
Quantity:
10 mg
Molecular Formula:
C25H27ClF4N2O4S
CAS:
1788071-27-1
Target:
Voltage-gated Sodium Channel Blockers
Purity:
0.98
Chemical Name or Material: __
Quantity: 100 μg
Molecular Formula: __
CAS: __
Target: __
Purity: __
Chemical Name or Material:
__
Quantity:
100 μg
Molecular Formula:
__
CAS:
__
Target:
__
Purity:
__
Chemical Name or Material: __
Quantity: 100 μg
Molecular Formula: __
CAS: __
Target: __
Purity: __
Chemical Name or Material:
__
Quantity:
100 μg
Molecular Formula:
__
CAS:
__
Target:
__
Purity:
__
Chemical Name or Material: __
Quantity: 100 μg
Molecular Formula: __
CAS: __
Target: __
Purity: __
Chemical Name or Material:
__
Quantity:
100 μg
Molecular Formula:
__
CAS:
__
Target:
__
Purity:
__