63-565

AT 1

Manufacturer: R&D Systems

CAS Number: 2098836-45-2

Select a Size

Pack Size SKU Availability Price
Each of 1 63-565-Each-of-1 In Stock ₹ 45,603.48

63-565 - Each of 1

₹ 45,603.48

In Stock

Quantity

1

Base Price: ₹ 45,603.48

GST (18%): ₹ 8,208.626

Total Price: ₹ 53,812.106

Chemical Name or Material

(2S,4R)-1-(2R)-2-Acetamido-3-[[6-[2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamido]hexyl]thio]-3-methylbutanoyl]-4-hydroxy-N-[4-(4-methylthiazol-5-yl)benzyl)pyrrolidinine-2-carboxamide

Assay Percent Range

>98%

Molecular Formula

C48H58ClN9O5S3

CAS

2098836-45-2

Quantity

5 mg

Formula Weight

Observed MW: 972.68

Other Options

Image Product Name Manufacturer Price Range
AX63069
2098836-45-2 | BRD4 Degrader AT1
A2B Chem ₹ 6,930.36 - ₹ 64,170.00

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Description

  • AT 1 is a cell penetrant Proteolysis Targeting Chimera (PROTAC®) compound based on (+)-JQ1 (Cat.No
  • 4499) conjugated to a von Hippel-Lindau (VHL) ligand
  • Rationally designed based on a ternary complex crystal structure to improve selectivity for BRD4 degradation compared to MZ1 (Cat.No
  • 6154)
  • Demonstrates profound and selective degradation of BRD4 in cells at 1-3 μM, with negligible loss of BRD2 and BRD3
  • PROTAC® is a registered trademark of Arvinas Operations, Inc., and is used under license

SAFETY INFORMATION

  • Recommended Storage : Store at -20°C

Compare Similar Items

Show Difference

Img

R&D Systems

63-565

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Chemical Name or Material:
(2S,4R)-1-(2R)-2-Acetamido-3-[[6-[2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamido]hexyl]thio]-3-methylbutanoyl]-4-hydroxy-N-[4-(4-methylthiazol-5-yl)benzyl)pyrrolidinine-2-carboxamide

Assay Percent Range:
>98%

Molecular Formula:
C48H58ClN9O5S3

CAS:
2098836-45-2

Quantity:
5 mg

Formula Weight:
Observed MW: 972.68

Img

eBioscience

63-571-182

--


Chemical Name or Material:
__

Assay Percent Range:
__

Molecular Formula:
__

CAS:
__

Quantity:
100 μg

Formula Weight:
__

Img

Fischer Scientific

63-572-5

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Chemical Name or Material:
(11β,16α)-16,17-[[(R)-Cyclohexylmethylene]bis(oxy)]-11-hydroxy-21-(2-methyl-1-oxopropoxy)pregna-1,4-diene-3,20-dione

Assay Percent Range:
>98%

Molecular Formula:
C32H44O7

CAS:
126544-47-6

Quantity:
25 mg

Formula Weight:
Observed MW: 540.7

Img

Fischer Scientific

63-575

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Chemical Name or Material:
(11β,16α)-16,17-[[(R)-Cyclohexylmethylene]bis(oxy)]-11-hydroxy-21-(2-methyl-1-oxopropoxy)pregna-1,4-diene-3,20-dione

Assay Percent Range:
>98%

Molecular Formula:
C32H44O7

CAS:
126544-47-6

Quantity:
5 mg

Formula Weight:
Observed MW: 540.7