7110842

Tocris Bioscience™ BX 430

Selective P2X4 allosteric antagonist

Manufacturer: Fischer Scientific

CAS Number: 688309-70-8

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Chemical Name or Material

N-[2,6-Dibromo-4-(1-methylethyl)phenyl]-N′-(3-pyridinyl)urea

Target

P2X Receptor Antagonists

Formula Weight

413.11

CAS

688309-70-8

Molecular Formula

C15H15Br2N3O

Purity

>99%

Other Options

Image Product Name Manufacturer Price Range
554550
Tocris Bioscience™ BX 430
Fischer Scientific ₹ 89,239.08
554510
Tocris Bioscience™ BX 430
Fischer Scientific ₹ 21,390.00
50-175-3030
Sigma Aldrich Fine Chemicals Biosciences BX430 >=98% (HPLC) | 688309-70-8 | MFCD02678819 | 25MG
Sigma Aldrich Fine Chemicals Biosciences ₹ 35,635.74
AH22890
688309-70-8 | BX 430
A2B Chem ₹ 1,368.96 - ₹ 10,181.64

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Description

  • Selective P2X4 allosteric antagonist (IC50 = 0.54 μM)
  • Exhibits >10-fold selectivity for human P2X4 receptors over P2X1, P2X2, P2X3, P2X5 and P2X7 receptors
  • Binds noncompetitively at extracellular allosteric site
  • Effective at human and zebrafish, but not mouse and rat P2X4 receptors.

SAFETY INFORMATION

  • Recommended Storage : Store at 4°C

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Selective P2X4 allosteric antagonis...


Chemical Name or Material:
N-[2,6-Dibromo-4-(1-methylethyl)phenyl]-N′-(3-pyridinyl)urea

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P2X Receptor Antagonists

Formula Weight:
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688309-70-8

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C15H15Br2N3O

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>99%

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