7110844

Tocris Bioscience™ Perlapine

Potent muscarinc DREADD agonist

Manufacturer: Fischer Scientific

CAS Number: 1977-11-3

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Chemical Name or Material

6-(4-Methyl-1-piperazinyl)-11 H-dibenz[b,e]azepine

Target

DREADD Activators

Formula Weight

291.39

CAS

1977-11-3

Molecular Formula

C19H21N3

Purity

99%

Other Options

Image Product Name Manufacturer Price Range
Tocris Bioscience™ Perlapine
-- ₹ 80,322.50
Tocris Bioscience™ Perlapine
-- ₹ 19,313.00
1977-11-3 | Perlapine
-- ₹ 4,628.00

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Description

  • Potent muscarinic DREADD agonist (pEC50 values are 8.38, 8.08 and 7.27 for hM1Dq, hM3Dq and hM4Di in vitro , respectively)
  • Exhibits >10,000-fold selectivity for hM3Dq over hM3 receptors.

SAFETY INFORMATION

  • Recommended Storage : Store at Room Temperature