7110891

Tocris Bioscience™ ML 382

MrgX1 (SNSR4) positive allosteric modulator

Manufacturer: Fischer Scientific

CAS Number: 1646499-97-9

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Chemical Name or Material

Mas-Related G Protein Coupled Receptor Modulators

Target

Sensory Neuron-Specific Receptor Agonists

Formula Weight

360.43

CAS

1646499-97-9

Molecular Formula

C18H20N2O4S

Purity

>98%

Other Options

Image Product Name Manufacturer Price Range
57-381-0
Tocris Bioscience™ ML 382
Fischer Scientific ₹ 18,460.43
57-385-0
Tocris Bioscience™ ML 382
Fischer Scientific ₹ 76,521.44
AX63168
1646499-97-9 | 2-(Cyclopropanesulfonamido)-N-(2-ethoxyphenyl)benzamide
A2B Chem ₹ 7,700.40 - ₹ 38,502.00

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Description

  • Selective MRGPRX1 positive allosteric modulator (EC50 = 190 nM)
  • Exhibits selectivity for MrgX1 over MrgX2, MrgC11 and a panel of 68 other GPCRs, ion channels and transporters
  • Enhances BAM (8-22) potency at MRGPRX1 by 7-fold.

SAFETY INFORMATION

  • Recommended Storage : Store at Room Temperature

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