7110906
Tocris Bioscience™ AZ 6102
Potent TNKS1/2 inhibitor
Manufacturer: Fischer Scientific
CAS Number: 1645286-75-4
The price for this product is unavailable. Please request a quote
Chemical Name or Material
rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
Target
Tankyrase Inhibitors
Formula Weight
428.53
CAS
1645286-75-4
Molecular Formula
C25H28N6O
Purity
>98%
Other Options
| Image | Product Name | Manufacturer | Price Range | |
|---|---|---|---|---|
 | Tocris Bioscience™ AZ 6102 | Fischer Scientific | ₹ 28,391.00 | |
| | Tocris Bioscience™ AZ 6102 | Fischer Scientific | ₹ 1,18,003.32 | |
 | eMolecules Medchem Express / AZ6102 / 5mg / 446262145 / HY-12975 / / 1645286-75-4 / MFCD28502279 / 428.540 / C25H28N6O | eMolecules | ₹ 9,825.60 | |
 | Sigma Aldrich Fine Chemicals Biosciences AZ6102 >=98% (HPLC) | 1645286-75-4 | 5MG | Sigma Aldrich Fine Chemicals Biosciences | ₹ 9,114.49 | |
| | Sigma Aldrich Fine Chemicals Biosciences AZ6102 >=98% (HPLC) | 1645286-75-4 | 25MG | Sigma Aldrich Fine Chemicals Biosciences | ₹ 36,850.45 | |
 | 4H-Pyrrolo[2,3-d]pyrimidin-4-one, 2-[4-[6-[(3R,5S)-3,5-dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-, rel- | Aaron Chemicals LLC | ₹ 10,947.00 - ₹ 1,04,753.00 | |
 | 1645286-75-4 | AZ6102 | A2B Chem | ₹ 3,026.00 - ₹ 42,186.00 |
Related Products
Description
- Potent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively)
- Exhibits >100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6
- Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM)
- Exhibits moderate oral bioavailability.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
Compare Similar Items
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Chemical Name or Material: rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
Target: Tankyrase Inhibitors
Formula Weight: 428.53
CAS: 1645286-75-4
Molecular Formula: C25H28N6O
Purity: >98%
Chemical Name or Material:
rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
Target:
Tankyrase Inhibitors
Formula Weight:
428.53
CAS:
1645286-75-4
Molecular Formula:
C25H28N6O
Purity:
>98%
Chemical Name or Material: N-5-Isoquinolinyl-N′-[[(4-(trifluoromethyl)phenyl]methyl]urea
Target: TRPV Antagonists
Formula Weight: 345.32
CAS: 581809-67-8
Molecular Formula: C18H14F3N3O
Purity: >98%
Chemical Name or Material:
N-5-Isoquinolinyl-N′-[[(4-(trifluoromethyl)phenyl]methyl]urea
Target:
TRPV Antagonists
Formula Weight:
345.32
CAS:
581809-67-8
Molecular Formula:
C18H14F3N3O
Purity:
>98%
Chemical Name or Material: 1,4-Dihydro-1′-[2-methyl-1H-benzimidazol-6-yl)carbonyl]-1-(1-methylethyl)-spiro[5H-indazole-5,4′-piperidin]-7(6H)-one
Target: Additional Lipid Metabolism Compounds
Formula Weight: 405.49
CAS: 1301214-47-0
Molecular Formula: C23H27N5O2
Purity: >98%
Chemical Name or Material:
1,4-Dihydro-1′-[2-methyl-1H-benzimidazol-6-yl)carbonyl]-1-(1-methylethyl)-spiro[5H-indazole-5,4′-piperidin]-7(6H)-one
Target:
Additional Lipid Metabolism Compounds
Formula Weight:
405.49
CAS:
1301214-47-0
Molecular Formula:
C23H27N5O2
Purity:
>98%
Chemical Name or Material: 5-(Dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-1,3-benzodiazole
Target: Bromodomain Inhibitors
Formula Weight: 488.62
CAS: 1962928-21-7
Molecular Formula: C29H36N4O3
Purity: >98%
Chemical Name or Material:
5-(Dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-1,3-benzodiazole
Target:
Bromodomain Inhibitors
Formula Weight:
488.62
CAS:
1962928-21-7
Molecular Formula:
C29H36N4O3
Purity:
>98%