73-521

Tocris™ YM 254890

Manufacturer: Tocris™

CAS Number: 568580-02-9

Select a Size

Pack Size SKU Availability Price
Each of 1 73-521-Each-of-1 In Stock ₹ 50,737.08

73-521 - Each of 1

₹ 50,737.08

In Stock

Quantity

1

Base Price: ₹ 50,737.08

GST (18%): ₹ 9,132.674

Total Price: ₹ 59,869.754

Chemical Name or Material

(R)-1-((3 S,6 S,9 S,12 S,18 R,21 S,22 R)-21-acetamido-18-benzyl-3-((R)-1-methoxyethyl)-4,9,10,12,16,22-hexamethyl-15-methylene-2,5,8,11,14,17,20-heptaoxo-1,19-dioxa-4,7,10,13,16-pentaazacyclodocosan-6-yl)-2-methylpropyl (2 S,3 R)-2-acetamido-3-hydroxy-4-methylpent

Quantity

1 mg

Molecular Formula

C46H69N7O15

CAS

568580-02-9

Target

GTPase Inhibitors

Purity

0.95

Other Options

Image Product Name Manufacturer Price Range
NC2316699
Cayman Chemical YM-254890 | 568580-02-9 | 960.1 g/mol | 1MG
Cayman Chemical ₹ 34,395.12
50-149-0016
AdipoGen YM-254890, 568580-02-9, 500mg
AdipoGen ₹ 19,678.80

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Description

  • YM 254890 is a Gα-protein inhibitor
  • Potently inhibits Gq/11 heterotrimeric G protein signaling
  • Inhibits ATP/UTP-induced Ca2+ increase in HCAE cells expressing P2Y2 receptor (IC50 = 50 nM); carbachol-induced production of IP1 in CHO cells expressing M1 receptor (IC50 = 95 nM); and ADP-induced Ca2+ increase in platelets, in vitro (IC50 = 2 μM)
  • Also inhibits Gs-induced cAMP elevation and G protein-coupled MAPK/ERK signaling.

SAFETY INFORMATION

  • Recommended Storage : Store at -20°C

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Show Difference

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Tocris™

73-521

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Chemical Name or Material:
(R)-1-((3 S,6 S,9 S,12 S,18 R,21 S,22 R)-21-acetamido-18-benzyl-3-((R)-1-methoxyethyl)-4,9,10,12,16,22-hexamethyl-15-methylene-2,5,8,11,14,17,20-heptaoxo-1,19-dioxa-4,7,10,13,16-pentaazacyclodocosan-6-yl)-2-methylpropyl (2 S,3 R)-2-acetamido-3-hydroxy-4-methylpent

Quantity:
1 mg

Molecular Formula:
C46H69N7O15

CAS:
568580-02-9

Target:
GTPase Inhibitors

Purity:
0.95

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5-(Acetylamino)-2-methyl-N-[(1 R)-1-(1-naphthalenyl)ethyl]benzamide

Quantity:
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Molecular Formula:
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Target:
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Purity:
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Chemical Name or Material:
N6-[(2-Propyn-1-yloxy)carbonyl]-L-lysine hydrochloride

Quantity:
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Molecular Formula:
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Target:
Unnatural Amino Acids

Purity:
0.95

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Chemical Name or Material:
N6-[(2-Propyn-1-yloxy)carbonyl]-L-lysine hydrochloride

Quantity:
50 mg

Molecular Formula:
C10H16N2O4.HCl

CAS:
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Target:
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Purity:
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