SML2203
SGC-GAK-1N
≥98% (HPLC)
Manufacturer: Sigma Aldrich
CAS Number: 2226517-74-2
Synonym(S): CA71, CA93 Negative Control, N-Methyl-6-(trifluoromethyl)-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine, SGC-GAK-1 Negative Control
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| 5 MG | SML2203-5-MG | In Stock | ₹ 9,850.75 |
| 25 MG | SML2203-25-MG | In Stock | ₹ 39,673.63 |
SML2203 - 5 MG
In Stock
Quantity
1
Base Price: ₹ 9,850.75
GST (18%): ₹ 1,773.135
Total Price: ₹ 11,623.885
Assay
≥98% (HPLC)
form
powder
color
dark green to black
solubility
DMSO: 2 mg/mL, clear
storage temp.
2-8°C
SMILES string
CN(C1=CC(OC)=C(OC)C(OC)=C1)C2=C3C(C=CC(C(F)(F)F)=C3)=NC=C2
Related Products
Description
- Biochem/physiol Actions: SGC-GAK-1N (CA71) is a structure analog of and the recommended negative control for the ATP-competitive cyclin G-associated kinase (GAK) inhibitor SGC-GAK-1 (CA93) (GAK KD = 1.9 nM/SGC-GAK-1 vs. 7.1 μM/SGC-GAK-1N by ligand competitive binding assay; GAK IC50 = 110 nM/SGC-GAK-1 vs. >50 μM/SGC-GAK-1N by cellular target engagement assay; Dengue viral entry and packaging IC50 = 920 nM/SGC-GAK-1 vs. >10 μM/SGC-GAK-1N). For characterization details of the active probe, SGC-GAK-1, please visit the SGC-GAK-1 probe summary on the Structural Genomics Consortium (SGC) website.SGC-GAK-1, the active probe, is available from Sigma. To learn more about and purchase SGC-GAK-1, click here.To learn about other SGC chemical probes, visit sigma.com/sgc
- Features and Benefits: SGC-GAK-1N is a negative control for SGC-GAK-1, a chemical probe available through a partnership with the Structural Genomics Consortium (SGC). To learn more and view other SGC chemical probes, visit sigma.com/SGC
SAFETY INFORMATION
WGK
WGK 3
Flash Point(F)
Not applicable
Flash Point(C)
Not applicable
Compare Similar Items
Show Difference
Assay: ≥98% (HPLC)
form: powder
color: dark green to black
solubility: DMSO: 2 mg/mL, clear
storage temp.: 2-8°C
SMILES string: CN(C1=CC(OC)=C(OC)C(OC)=C1)C2=C3C(C=CC(C(F)(F)F)=C3)=NC=C2
Assay:
≥98% (HPLC)
form:
powder
color:
dark green to black
solubility:
DMSO: 2 mg/mL, clear
storage temp.:
2-8°C
SMILES string:
CN(C1=CC(OC)=C(OC)C(OC)=C1)C2=C3C(C=CC(C(F)(F)F)=C3)=NC=C2
Assay: ≥98% (HPLC)
form: powder
color: white to beige
solubility: DMSO: 2 mg/mL, clear
storage temp.: 2-8°C
SMILES string: ClC1=CC(S(N2CCC(C(NCC3=CC=C(F)C=C3)=O)CC2)(=O)=O)=CC(Cl)=C1
Assay:
≥98% (HPLC)
form:
powder
color:
white to beige
solubility:
DMSO: 2 mg/mL, clear
storage temp.:
2-8°C
SMILES string:
ClC1=CC(S(N2CCC(C(NCC3=CC=C(F)C=C3)=O)CC2)(=O)=O)=CC(Cl)=C1
Assay: ≥98% (HPLC)
form: powder
color: white to beige
solubility: DMSO: 2 mg/mL, clear
storage temp.: 2-8°C
SMILES string: CCN(CC)S(NC1=CC=CC(C2=CC(NN=C3NC(C4CC4)=O)=C3C=C2)=C1)(=O)=O
Assay:
≥98% (HPLC)
form:
powder
color:
white to beige
solubility:
DMSO: 2 mg/mL, clear
storage temp.:
2-8°C
SMILES string:
CCN(CC)S(NC1=CC=CC(C2=CC(NN=C3NC(C4CC4)=O)=C3C=C2)=C1)(=O)=O
Assay: ≥98% (HPLC)
form: powder
color: white to beige
solubility: DMSO: 2 mg/mL, clear
storage temp.: 2-8°C
SMILES string: O=C(C(C)C)NC1=NNC2=C1C=CC(C3=CC(NS(C4CC4)(=O)=O)=CC=C3)=C2
Assay:
≥98% (HPLC)
form:
powder
color:
white to beige
solubility:
DMSO: 2 mg/mL, clear
storage temp.:
2-8°C
SMILES string:
O=C(C(C)C)NC1=NNC2=C1C=CC(C3=CC(NS(C4CC4)(=O)=O)=CC=C3)=C2