60-051-0

Tocris Bioscience™ PF 3758309 dihydrochloride

Manufacturer: Fischer Scientific

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Pack Size SKU Availability Price
Each of 1 60-051-0-Each-of-1 In Stock ₹ 11,512.95

60-051-0 - Each of 1

₹ 11,512.95

In Stock

Quantity

1

Base Price: ₹ 11,512.95

GST (18%): ₹ 2,072.331

Total Price: ₹ 13,585.281

Chemical Name or Material

PF 3758309 Dihydrochloride

Quantity

10 mg

Molecular Formula

C25H30N8OS.2HCl

Physical Form

Solid

Product Type

Bioactive Small Molecule

Synonym

N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide dihydrochloride

Solubility

Soluble to 100mM in water and to 100mM in DMSO

Formula Weight

563.55

Color

Off-white

Purity

>98%

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Description

  • Potent PAK4 inhibitor (IC50 = 1.3 nM; Kd = 2.7 nM)
  • Inhibits proliferation and anchorage-independent growth of a panel of tumor cell lines in vitro
  • Suppresses growth of human HCT116 and A549 tumor cell xenografts in mice
  • Orally available.

SAFETY INFORMATION

  • Recommended Storage : Store at -20°C

Compare Similar Items

Show Difference

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Fischer Scientific

60-051-0

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Chemical Name or Material:
PF 3758309 Dihydrochloride

Quantity:
10 mg

Molecular Formula:
C25H30N8OS.2HCl

Physical Form:
Solid

Product Type:
Bioactive Small Molecule

Synonym:
N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide dihydrochloride

Solubility:
Soluble to 100mM in water and to 100mM in DMSO

Formula Weight:
563.55

Color:
Off-white

Purity:
>98%

Img

Fischer Scientific

60-055-0

--


Chemical Name or Material:
PF 3758309 Dihydrochloride

Quantity:
50 mg

Molecular Formula:
C25H30N8OS.2HCl

Physical Form:
Solid

Product Type:
Bioactive Small Molecule

Synonym:
N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide dihydrochloride

Solubility:
Soluble to 100mM in water and to 100mM in DMSO

Formula Weight:
563.55

Color:
Off-white

Purity:
>98%

Img

Fischer Scientific

60-081-0

--


Chemical Name or Material:
TP 064

Quantity:
10 mg

Molecular Formula:
C28H34N4O2

Physical Form:
Solid

Product Type:
Bioactive Small Molecule

Synonym:
N-Methyl-N-((2-(1-(2-(methylamino)ethyl)piperidin-4-yl)pyridin-4-yl)methyl)-3-phenoxybenzamide

Solubility:
Soluble to 100mM in 1eq. HCl and to 100mM in DMSO

Formula Weight:
458.6

Color:
White

Purity:
>98%

Img

Fischer Scientific

60-085-0

--


Chemical Name or Material:
TP 064

Quantity:
50 mg

Molecular Formula:
C28H34N4O2

Physical Form:
Solid

Product Type:
Bioactive Small Molecule

Synonym:
N-Methyl-N-((2-(1-(2-(methylamino)ethyl)piperidin-4-yl)pyridin-4-yl)methyl)-3-phenoxybenzamide

Solubility:
Soluble to 100mM in 1eq. HCl and to 100mM in DMSO

Formula Weight:
458.6

Color:
White

Purity:
>98%