71-575

Tocris Bioscience™ YKL 5-124

Manufacturer: Tocris Bioscience™

CAS Number: 1957203-01-8

Select a Size

Pack Size SKU Availability Price
Each of 1 71-575-Each-of-1 In Stock ₹ 31,999.44

71-575 - Each of 1

₹ 31,999.44

In Stock

Quantity

1

Base Price: ₹ 31,999.44

GST (18%): ₹ 5,759.899

Total Price: ₹ 37,759.339

Chemical Name or Material

N-[(1 S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[[4-[(1-oxo-2-propen-1-yl)amino]benzoyl]amino]pyrrolo[3,4-c]pyrazole-5(1 H)-carboxamide

Quantity

5 mg

Molecular Formula

C28H33N7O3

CAS

1957203-01-8

Target

Cyclin-dependent Kinase Inhibitors

Purity

0.95

Other Options

Image Product Name Manufacturer Price Range
50-226-0395
Medchemexpress LLC HY-101257 10mg , YKL-5-124 CAS:1957203-01-8 Purity:>98%
Medchemexpress LLC ₹ 39,079.53
50-226-0396
Medchemexpress LLC HY-101257 25mg , YKL-5-124 CAS:1957203-01-8 Purity:>98%
Medchemexpress LLC ₹ 62,527.25
50-225-9879
Medchemexpress LLC HY-101257 5mg , YKL-5-124 CAS:1957203-01-8 Purity:>98%
Medchemexpress LLC ₹ 22,908.69
BG26438
1957203-01-8 | YKL-5-124
A2B Chem ₹ 11,550.60 - ₹ 87,613.44

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Description

  • YKL-5-124 is a potent and selective CDK7/Mat1/CycH and cyclin dependent kinase (CDK7) inhibitor (IC50 values = 9.7 nM and 53.5 nM, respectively)
  • YKL-5-124 shows 100-fold selectivity over CDK9 and CDK2
  • YKL-5-124 induces cell cycle arrest at the G1/S transition, inhibits E2F-driven gene expression and inhibits CDK1 and CDK3 T-loop phosphorylation.

SAFETY INFORMATION

  • Recommended Storage : Store at -20°C

Compare Similar Items

Show Difference

Img

Tocris Bioscience™

71-575

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Chemical Name or Material:
N-[(1 S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[[4-[(1-oxo-2-propen-1-yl)amino]benzoyl]amino]pyrrolo[3,4-c]pyrazole-5(1 H)-carboxamide

Quantity:
5 mg

Molecular Formula:
C28H33N7O3

CAS:
1957203-01-8

Target:
Cyclin-dependent Kinase Inhibitors

Purity:
0.95

Img

MilliporeSigma™

71-590-3MI

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Chemical Name or Material:
__

Quantity:
100 μg

Molecular Formula:
__

CAS:
__

Target:
__

Purity:
__

Img

MilliporeSigma™

71-591-3MI

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Chemical Name or Material:
__

Quantity:
75 μL

Molecular Formula:
__

CAS:
__

Target:
__

Purity:
__

Img

Tocris™

71-605

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Chemical Name or Material:
4-(1,1-Dimethylethyl)-N-[3-[6-[[4-[[4-[6-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1 H-isoindol-4-yl]amino]acetyl]amino]hexyl]-1-piperazinyl]carbonyl]phenyl]amino]-4,5-dihydro-4-methyl-5-oxo-2-pyrazinyl]-2-methylphenyl]benzamide

Quantity:
5 mg

Molecular Formula:
C55H62N10O8

CAS:
2366132-45-6

Target:
Active Degraders

Purity:
0.98