7161659

Tocris Bioscience™ Pelitinib

Potent and irreversible EGFR inhibitor (IC50 = 20-80 nM); orally bioavailable

Manufacturer: Fischer Scientific

CAS Number: 257933-82-7

The price for this product is unavailable. Please request a quote

Chemical Name or Material

(2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide

Synonym

EKB-569

Formula Weight

467.92

CAS

257933-82-7

Molecular Formula

C24H23ClFN5O2

Purity

97%

Other Options

Image Product Name Manufacturer Price Range
63-492-5
Tocris Bioscience™ Pelitinib
Fischer Scientific ₹ 42,776.58
63-495
Tocris Bioscience™ Pelitinib
Fischer Scientific ₹ 11,115.96
50-186-5651
Sigma Aldrich Fine Chemicals Biosciences Pelitinib >=98% (HPLC) | 257933-82-7 | 25MG
Sigma Aldrich Fine Chemicals Biosciences ₹ 61,687.05
50-801-8
Selleck Chemical LLC Pelitinib (EKB-569) 5mg 257933-82-7
Selleck Chemical LLC ₹ 15,400.80
50-801-9
Selleck Chemical LLC Pelitinib (EKB-569) 25mg 257933-82-7
Selleck Chemical LLC ₹ 47,451.58
AD54879
257933-82-7 | Pelitinib
A2B Chem ₹ 2,823.48 - ₹ 1,50,585.60

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Description

  • Selective for EGFR over Src, MEK/ERK, erbB2, Raf, c-Met and Cdk4 (IC50 values are 282, 800, 1255, 3353, 4100 and >20,000) Inhibits the growth of tumors overexpressing EGFR in vivo Orally bioavailable

SAFETY INFORMATION

  • Recommended Storage : Store at -20°C

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Chemical Name or Material:
(2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide

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C24H23ClFN5O2

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