7166780
Tocris™ GSK 1016790A
Potent TRPV4 agonist
Manufacturer: Fischer Scientific
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Molecular Formula
C28H32Cl2N4O6S2
Formula Weight
655.61
Product Type
Agonist
Purity
98%
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Description
- Description GSK 1016790A is a potent TRPV4 agonist; elicits Ca2+ influx in human and mouse TRPV4-expressing HEK cells (EC50 values of 2.1 and 18 nM, respectively)
- Enhances insulin mRNA expression
- Increases ERK1/2 phosphorylation and NO production
- Exhibits no activity at TRPM8 and TRPA1 (20 μM) channels
- Induces bladder overactivity in TRPV4+/+ mice.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
Compare Similar Items
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Molecular Formula: C28H32Cl2N4O6S2
Formula Weight: 655.61
Product Type: Agonist
Purity: 98%
Molecular Formula:
C28H32Cl2N4O6S2
Formula Weight:
655.61
Product Type:
Agonist
Purity:
98%
Molecular Formula: C27H40N4O3.HCl
Formula Weight: 505.09
Product Type: Antagonist
Purity: 98%
Molecular Formula:
C27H40N4O3.HCl
Formula Weight:
505.09
Product Type:
Antagonist
Purity:
98%
Molecular Formula: C33H25NO8Na2
Formula Weight: 609.54
Product Type: Antagonist
Purity: 98%
Molecular Formula:
C33H25NO8Na2
Formula Weight:
609.54
Product Type:
Antagonist
Purity:
98%
Molecular Formula: C18H16FN3O
Formula Weight: 309.34
Product Type: Inhibitor
Purity: 98%
Molecular Formula:
C18H16FN3O
Formula Weight:
309.34
Product Type:
Inhibitor
Purity:
98%