72-855
Tocris Bioscience™ DCLK1-IN-1
Manufacturer: Tocris Bioscience™
CAS Number: 2222635-15-4
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 72-855-Each-of-1 | In Stock | ₹ 26,095.80 |
72-855 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 26,095.80
GST (18%): ₹ 4,697.244
Total Price: ₹ 30,793.044
Chemical Name or Material
5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6 H-pyrimido[4,5-b][1,4 ]benzodiazepin-6-one
Quantity
5 mg
Molecular Formula
C26H28F3N7O2
CAS
2222635-15-4
Target
Other Kinase Inhibitors
Purity
0.98
Other Options
| Image | Product Name | Manufacturer | Price Range | |
|---|---|---|---|---|
 | eMolecules Medchem Express / DCLK1-IN-1 / 5mg / 532149305 / HY-135985 / / 2222635-15-4 / [null] / 527.552 / C26H28F3N7O2 | eMolecules | ₹ 35,264.41 | |
 | 2222635-15-4 | 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one | A2B Chem | ₹ 4,106.88 - ₹ 2,46,498.36 |
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Description
- DCLK1-IN-1 is a potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor (IC50 values are DCLK1 =9.5 and 57.2 nM and DCLK2 = 31 and 103 nM in binding and kinase assay, respectively)
- Exhibits no significant activity against ERK5, ACK, BRD4 and LRRK2
- Exhibits DCLK inhibition in pancreatic ductal adenocarcinoma (PDAC) organoid models
- Orally bioavailable.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
Compare Similar Items
Show Difference
Chemical Name or Material: 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6 H-pyrimido[4,5-b][1,4 ]benzodiazepin-6-one
Quantity: 5 mg
Molecular Formula: C26H28F3N7O2
CAS: 2222635-15-4
Target: Other Kinase Inhibitors
Purity: 0.98
Chemical Name or Material:
5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6 H-pyrimido[4,5-b][1,4 ]benzodiazepin-6-one
Quantity:
5 mg
Molecular Formula:
C26H28F3N7O2
CAS:
2222635-15-4
Target:
Other Kinase Inhibitors
Purity:
0.98
Chemical Name or Material: __
Quantity: 1 mg
Molecular Formula: C71H84N10O25
CAS: __
Target: Other Fluorescent Probes
Purity: 0.95
Chemical Name or Material:
__
Quantity:
1 mg
Molecular Formula:
C71H84N10O25
CAS:
__
Target:
Other Fluorescent Probes
Purity:
0.95
Chemical Name or Material: (2 aR,5 aR,6 S,6 aR,8 R,9 aR,10 AS,10 bR,10 cR)-8-(3-Furanyl)-2 A,5 A,6,6 A,8,9,9 A,10 A,10 b,10 c-decahydro-2 A,5 A,6 A,7-tetramethyl-2,5-dioxo-2 H,5 H-cyclopenta[d']naphtho[1,8-bc:2,3-b']difuran-6-acetic acid methyl ester
Quantity: 25 mg
Molecular Formula: C27H30O7
CAS: 25990-37-8
Target: Ubiquitin Ligase (E3) Inhibitors
Purity: 0.97
Chemical Name or Material:
(2 aR,5 aR,6 S,6 aR,8 R,9 aR,10 AS,10 bR,10 cR)-8-(3-Furanyl)-2 A,5 A,6,6 A,8,9,9 A,10 A,10 b,10 c-decahydro-2 A,5 A,6 A,7-tetramethyl-2,5-dioxo-2 H,5 H-cyclopenta[d']naphtho[1,8-bc:2,3-b']difuran-6-acetic acid methyl ester
Quantity:
25 mg
Molecular Formula:
C27H30O7
CAS:
25990-37-8
Target:
Ubiquitin Ligase (E3) Inhibitors
Purity:
0.97
Chemical Name or Material: (2 aR,5 aR,6 S,6 aR,8 R,9 aR,10 AS,10 bR,10 cR)-8-(3-Furanyl)-2 A,5 A,6,6 A,8,9,9 A,10 A,10 b,10 c-decahydro-2 A,5 A,6 A,7-tetramethyl-2,5-dioxo-2 H,5 H-cyclopenta[d']naphtho[1,8-bc:2,3-b']difuran-6-acetic acid methyl ester
Quantity: 5 mg
Molecular Formula: C27H30O7
CAS: 25990-37-8
Target: Ubiquitin Ligase (E3) Inhibitors
Purity: 0.97
Chemical Name or Material:
(2 aR,5 aR,6 S,6 aR,8 R,9 aR,10 AS,10 bR,10 cR)-8-(3-Furanyl)-2 A,5 A,6,6 A,8,9,9 A,10 A,10 b,10 c-decahydro-2 A,5 A,6 A,7-tetramethyl-2,5-dioxo-2 H,5 H-cyclopenta[d']naphtho[1,8-bc:2,3-b']difuran-6-acetic acid methyl ester
Quantity:
5 mg
Molecular Formula:
C27H30O7
CAS:
25990-37-8
Target:
Ubiquitin Ligase (E3) Inhibitors
Purity:
0.97