7235824
Tocris™ VCP 171
Positive allosteric modulator (PAM) of A1 receptors; also allosteric partial agonist in absence of orthosteric agonist
Manufacturer: Fischer Scientific
CAS Number: 1018830-99-3
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Chemical Name or Material
[2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenylmethanone
Target
Adenosine A1 Receptor Modulators
Purity
0.98
CAS
1018830-99-3
Molecular Formula
C18H12F3NOS
Other Options
| Image | Product Name | Manufacturer | Price Range | |
|---|---|---|---|---|
 | Tocris™ VCP 171 | Fischer Scientific | ₹ 20,842.42 | |
| | Tocris™ VCP 171 | Fischer Scientific | ₹ 87,835.90 |
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Description
- VCP 171 is an adenosine A1 receptor positive allosteric modulator (PAM) (pKB = 5.65, binding cooperativity with NECA 0.68)
- In absence of orthosteric agonist, VCP171 behaves as an allosteric partial agonist, inhibiting cAMP activity
- Inhibits AMPA receptor-mediated evoked excitatory postsynaptic current (eEPSC) amplitude in lamina I and II neurons in a rat partial nerve-injury model of neuropathic pain.
SAFETY INFORMATION
- Recommended Storage : Store at -20°C
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Chemical Name or Material: [2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenylmethanone
Target: Adenosine A1 Receptor Modulators
Purity: 0.98
CAS: 1018830-99-3
Molecular Formula: C18H12F3NOS
Chemical Name or Material:
[2-Amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenylmethanone
Target:
Adenosine A1 Receptor Modulators
Purity:
0.98
CAS:
1018830-99-3
Molecular Formula:
C18H12F3NOS
Chemical Name or Material: N-[(1 S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5 H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide hydrochloride
Target: NPY Receptor Antagonists
Purity: 0.98
CAS: 2624332-04-1
Molecular Formula: C49H57N11O6.HCl
Chemical Name or Material:
N-[(1 S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5 H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide hydrochloride
Target:
NPY Receptor Antagonists
Purity:
0.98
CAS:
2624332-04-1
Molecular Formula:
C49H57N11O6.HCl
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