77-572
Tocris Bioscience™ AZ 13824374
Manufacturer: Tocris Bioscience™
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| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 77-572-Each-of-1 | In Stock | ₹ 34,538.86 |
77-572 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 34,538.86
GST (18%): ₹ 6,216.995
Total Price: ₹ 40,755.855
Chemical Name or Material
(1R,2R,5S)-11-(8-((1-(2-Fluoro-2-methylpropyl)piperidin-4-yl)amino)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine-6-carbonyl)-2-isopropyl-2,3,5,6-tetrahydro-1,5-epiminobenzo[d]azocin-4(1H)-one
Quantity
2 mg
Target
ATAD2
Molecular Formula
C30H39FN8O2
Related Products
Description
- AZ 13824374 is a potent and selective inhibitor of ATPase family AAA domain-containing protein 2 (ATAD2) bromodomain (pIC50 values are 6.2 and 8.2 in NanoBRET assay and FRET assay, respectively)
- It is >100-fold selective over a range of epigenetic targets from ROMO scan panel (DiscoveRx Corp.)
- AZ 13824374 shows cellular target engagement (cellular inhibition pIC50 = 6.9) and antiproliferative activity in a range of breast cancer cell lines.
SAFETY INFORMATION
- Recommended Storage : Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date.
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Chemical Name or Material: (1R,2R,5S)-11-(8-((1-(2-Fluoro-2-methylpropyl)piperidin-4-yl)amino)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine-6-carbonyl)-2-isopropyl-2,3,5,6-tetrahydro-1,5-epiminobenzo[d]azocin-4(1H)-one
Quantity: 2 mg
Target: ATAD2
Molecular Formula: C30H39FN8O2
Chemical Name or Material:
(1R,2R,5S)-11-(8-((1-(2-Fluoro-2-methylpropyl)piperidin-4-yl)amino)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazine-6-carbonyl)-2-isopropyl-2,3,5,6-tetrahydro-1,5-epiminobenzo[d]azocin-4(1H)-one
Quantity:
2 mg
Target:
ATAD2
Molecular Formula:
C30H39FN8O2
Chemical Name or Material: -3-[[[(2 S,4 R)-1-[-2-(1-Fluorocyclopropan-1-ylcarbonylamino)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidin-2-yl]carbonyl]amino]-3-[4-(4-methylthiazol-5-yl)phenyl]propanoic acid
Quantity: 50 mg
Target: Degrader Building Blocks
Molecular Formula: C28H35FN4O6S
Chemical Name or Material:
-3-[[[(2 S,4 R)-1-[-2-(1-Fluorocyclopropan-1-ylcarbonylamino)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidin-2-yl]carbonyl]amino]-3-[4-(4-methylthiazol-5-yl)phenyl]propanoic acid
Quantity:
50 mg
Target:
Degrader Building Blocks
Molecular Formula:
C28H35FN4O6S
Chemical Name or Material: 4-[[2,5-Bis[[4-(1-pyrrolidinyl)-1-piperidinyl]carbonyl]phenyl]amino]benzoic acid ditrifluoroacetate
Quantity: 50 mg
Target: Degrader Building Blocks
Molecular Formula: C33H43N5O4.2CF3CO2H
Chemical Name or Material:
4-[[2,5-Bis[[4-(1-pyrrolidinyl)-1-piperidinyl]carbonyl]phenyl]amino]benzoic acid ditrifluoroacetate
Quantity:
50 mg
Target:
Degrader Building Blocks
Molecular Formula:
C33H43N5O4.2CF3CO2H
Chemical Name or Material: Surfactants-MBAS QC Sample
Quantity: 10 mL
Target: __
Molecular Formula: __
Chemical Name or Material:
Surfactants-MBAS QC Sample
Quantity:
10 mL
Target:
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Molecular Formula:
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